Preserved supervised synthesis

Leuprolide synthesis · version 1

This URL preserves the exact reviewed public wording and source set for synthesis version 1.

Supervised synthesis

What do selected human studies report about Leuprolide?

Manually reviewed August 19, 2026 · version 1

Browse all Human Evidence Reviews · Open preserved synthesis version 1 →

A bounded review of two randomized comparisons involving leuprolide: one pelvic-pain trial and one androgen-deprivation trial using leuprolide as the active comparator.12

Bottom line from this bounded source set

In the reviewed pelvic-pain trial, both treatment groups improved without a significant between-group difference. In the prostate-cancer trial, the oral comparator produced more sustained testosterone suppression than leuprolide; that biochemical endpoint does not establish a difference in cancer survival.12

Reviewed study record

Endometriosis-associated pelvic-pain trial

Design

A prospective, randomized, double-blind controlled trial compared leuprolide with continuous oral contraceptives over 48 weeks.1

Population

The trial enrolled 47 women with endometriosis-associated pelvic pain at academic medical centers in two U.S. cities.1

Outcomes reported

Pain and depression scores declined significantly from baseline in both groups, while the reported reductions did not differ significantly between groups.1

Limitations

The trial was small, and improvement within each group does not establish that the treatments were equivalent across broader populations or longer follow-up.1

Reviewed study record

HERO androgen-deprivation trial

Design

A sponsor-funded, randomized Phase 3 trial compared oral relugolix with leuprolide for 48 weeks; sustained testosterone suppression was the primary endpoint.2

Population

The trial randomized 930 men with advanced prostate cancer, including 308 assigned to leuprolide.2

Outcomes reported

Sustained testosterone suppression was reported for 96.7% of the relugolix group and 88.8% of the leuprolide group, meeting the trial's noninferiority and superiority criteria for that endpoint.2

Limitations

Leuprolide was the comparator, not the experimental treatment, and the primary result concerned testosterone suppression rather than cancer progression or survival.2

Reviewed source set

  1. PubMed · 21300339Randomized trial of leuprolide versus continuous oral contraceptives in the treatment of endometriosis-associated pelvic pain ↗PubMed PMID 21300339 · EFetch XML reviewed 2026-08-19 · payload SHA-256 acdc72872e6bd7de45be01788dfd401b16780ce2ac46cd3834a9299cbf8314c3
    No registered Crossref update in the reviewed snapshotChecked August 19, 2026 for DOI 10.1016/j.fertnstert.2011.01.027. This bounded result is not proof that the publication has never been corrected or retracted. Open the pinned Crossref work endpoint ↗
  2. PubMed · 32469183Oral Relugolix for Androgen-Deprivation Therapy in Advanced Prostate Cancer ↗PubMed PMID 32469183 · EFetch XML reviewed 2026-08-19 · payload SHA-256 ff23e8f570d660744b13fbe1420af8f24b062e1dad2ce2b36eee4e240dd2a36b
    No registered Crossref update in the reviewed snapshotChecked August 19, 2026 for DOI 10.1056/nejmoa2004325. This bounded result is not proof that the publication has never been corrected or retracted. Open the pinned Crossref work endpoint ↗